O paipa a le Laboratory

Oloa

Pimobendan 74150-27-9 Metabolism PDE inhibitor

Fa'amatalaga Puupuu:

igoa ole oloa:Pimobendan
upu uiga tutusa:4,5-Dihydro-6-[2-(4-methoxyphenyl)-1H-benzimidazol-6-yl]-5-methyl-3(2H)-pyridazinone
Numera CAS:74150-27-9
Tulaga lelei:USP43
fua mole:C19H18N4O2
mamafa mole:334.37


Fa'amatalaga Oloa

Faailoga o oloa

Totogi:T/T, L/C
Puna'oa:Saina
Taulaga Va'a:Beijing/Shanghai/Hangzhou
Poloaiga (MOQ):1g
Taimi muamua:3 aso faigaluega
Gaosi gaosiga:1kg/masina
Tulaga teuina:Teu i totonu o se nofoaga malulu, matutu, potu vevela.
Mea fa'apipi'i:fagu, fagu
Tele le afifi:1g/ fagu, 5/ fagu, 10g/ fagu, 50g/fagu, 500g/fagu
Fa'amatalaga saogalemu:UN 2811 6.1/PG 3

Pimobendan

Folasaga

Pimobendan, o se vaila'au fa'afoma'i.O se faʻamaʻi maʻaleʻale calcium ma se inhibitor filifilia o le phosphodiesterase 3 (PDE3) faʻatasi ai ma aʻafiaga lelei inotropic ma vasodilator.

O le Pimobendan e fa'aaogaina i le puleaina o le faaletonu o le fatu i taifau, e masani ona mafua mai i le myxomatous mitral valve maʻi (lea na taʻua muamua o le endocardiosis), poʻo le cardiomyopathy dilated.O suʻesuʻega ua faʻaalia e pei o le monotherapy, o le pimobendan e faʻateleina ai le taimi e ola ai ma faʻaleleia le lelei o le olaga i tagata gasegase e maua i le fatu faʻaletonu lona lua i le faʻamaʻi valve mitral pe a faʻatusatusa i le benazepril, o le ACE inhibitor.

Fa'amatalaga (USP43)

Aitema

Fa'amatalaga

Fa'aaliga

Pa'epa'e pe lanu samasama pa'epa'e, hygroscopic

Mp

E tusa o le 242℃

Solubility

E le mafai ona solu ile vai, solu fua ile dimethylformamide, solute laititi ile acetone ma le methanil.

Fa'ailoaga

Infrared absorption spectrophotometry, Fa'atusatusaga pimobendan CRS.

O le taimi fa'atumauina o le tumutumu tele o le Sample solution e fetaui ma le fa'ata'ita'iga o fa'atauga masani, e pei ona maua i le su'ega Organic Impurities.

Metala mamafa

≤10ppm

Fa'amamafa

P90 ≤ 25μm

Lapopo'a o vaega

20-80 mata

Solivai totoe

≤ 500ppm

Vai

≤ 1.0%

Su'ega

98.0%~102.0%

Lefulefu sulphated

≤ 0.10%

Mea fa'atatau (HPLC)

le mama A

≤ 0.10%

le mama B

≤ 0.10%

So'o se isi mea leaga

≤ 0.10%

Le mama atoatoa

≤ 0.20%


  • Muamua:
  • Sosoo ai: