Mirabegron 223673-61-8 Inhibitor Neuronal signal
Totogi:T/T, L/C
Puna'oa:Saina
Taulaga Va'a:Beijing/Shanghai/Hangzhou
Gaosi gaosiga:100kg/masina
Poloaiga(MOQ):25kg
Taimi muamua:3 Aso Galue
Tulaga teuina:Teu i totonu o se nofoaga malulu, matutu, potu vevela.
Mea fa'apipi'i:talipalau
Tele le afifi:25kg/tapa
Fa'amatalaga saogalemu:E le o ni oloa matautia

Folasaga
Mirabegron, o se beta-3 adrenergic receptor agonist, lea e faaosofia ai le beta-3 adrenergic receptor ma faʻamalieina le musele lamolemole detrusor, ma faʻapupulaina ai le mana o le vevela ma faʻaaogaina e togafitia ai faʻamaoniga o le manava malosi (OAB), e pei o le faʻamalosi, faanatinati, ma le tele o taimi.
O ona faʻamanuiaga e tutusa ma vailaʻau antimuscarinic e pei o le solifenacin poʻo le tolterodine.
Fa'amatalaga (USP/EP)
Aitema | Fa'amatalaga |
Fa'aaliga | Pa'epa'e e pa'epa'e pa'epa'e |
Fa'ailoaga | IR, HPLC |
vai vai | NMT 0.5% |
Toega ile mu | NMT 0.1% |
Uamea mamafa | NMT 20ppm |
Palladium anotusi | NMT 20ppm |
Optical isomer | NTM 0.5% |
Mea fa'atatau | Z-168*: NMT 0.15% |
SC03610*: NMT 0.15% | |
So'o se isi mea leaga e le iloa: NMT 0.10% | |
Aofa'i le mama: NMT 0.5% | |
2-(2-aminothianzol-4-yl) acetic acid | NMT 0.1% |
Solitu totoe | Methanol: NMT 0.3% |
Ethyl acetate: NMT 0.5% | |
THF: NMT 0.072% | |
Pesini: NMT 0.0002% | |
Toluene: NMT 0.089% | |
Su'ega | 98.0% - 102.0% |
PSD | D (0.5): 10μm - 30μm |
D (0.9): 20μm - 80μm |